產品簡介

天津益元利康科技有限公司是Macrocyclics代理
Macrocyclics 由A. Dean Sherry教授于1995年創立。公司提供廣泛的目錄產品庫，旨在基礎和應用層面滿足研究客戶的需求，以及定制 cGMP 產品和服務，以加快早期臨床開發計劃。產品包括廣泛的雙功能配體系列，專為與單克隆抗體和肽片段結合而設計的生物靶向。

雙功能螯合劑（BFCs）

B-277

2-Aminoethyl-mono-amide-DOTA-tris(t-Bu ester)

173308-19-5

1,4,7,10-Tetraazacyclododecane-1,4,7-tris(t-butyl-acetate)-10-(aminoethylacetamide)

B-259

4-Aminobutyl-DOTA

753421-63-5

1,4,7,10-Tetraazacyclododecane-1,4,7-tris(acetic   acid)-10-(4-aminobutyl)acetamide

B-279

4-Aminobutyl-DOTA-tris (t-butyl ester)

1402393-59-2

1,4,7,10-Tetraazacyclododecane-1,4,7-tris(t-butyl   acetate)-10-(4-aminobutyl)acetamide

B-288

Azido-mono-amide-DOTA

1227407-76-2

1,4,7,10-Tetraazacyclododecane-1,4,7-tris(acetic   acid)-10-(azidopropyl ethylacetamide)

共軛物

C-210

DO3A-Serotonin

2125661-93-8

1-(5-Hydroxyindole-3-ethylacetamide)-4,7,10-triacetic   acid-1,4,7,10-tetraazacyclododecane

C-100

DOTA-Biotin-Sarcosine

180978-54-5

(N-methyl-N-(hexahydro-2-oxo-1H-thieno[3,4-d]-imidazol-4-yl)-oxopentyl)glycyl-2-(S)-(4-aminobenzyl)-1,4,7,10-tetraacetic   acid-1,4,7,10-tetraazacyclododecane

C-220

DOTATATE

177943-89-4

DOTA-d-Phe-Cys-Tyr-d-Trp-Lys-Thr-Cys-Thr

熒光探針

D-100

EAM-1

287970-46-1

N,N,N-Trimethyl-2[(7-nitro-1,2,3-benzoxadiazol-4-yl)amino]   ethanaminium iodide

D-110

EAM-2

2125661-97-2

N,N-Dimethyl-N-(2-hydroxyethyl)-2[(7-nitro-1,2,3-benzoxadiazol-4-yl)amino]   ethanaminium bromide

大環配體

M-200

CB-Cyclam

130701-19-8

1,4,8,11-Tetraazabicyclo[6.6.2]hexadecane

M-220

CB-TE2A

313229-90-2

1,4,8,11-Tetraazabicyclo[6.6.2]hexadecane-4,11-diacetic   acid

M-100

Cyclen

294-90-6

1,4,7,10-Tetraazacyclododecane

M-190

DiAmSar

91002-72-1

1,8-Diamino-3,6,10,13,16,19-hexaazabicyclo[6,6,6]-eicosane

M-125

DO2A

112193-75-6

1,4,7,10-Tetraazacyclododecane-1,7-diacetic acid

磁共振試劑

M-503

Eu-DOTA-4AmC

481668-57-9

Europium (III) 1,4,7,10-Tetraazacyclododecane-1,4,7,10-tetrakis(acetamidoacetic   acid)

X-287

Gd-DO3A-Butylamine

782423-00-1

Gadolinium (III)   1,4,7,10-Tetraazacyclododecane-1,4,7-tris(acetic   acid)-10-(4-aminobutyl)acetamide

M-147

Gd-DOTA

72573-82-1

Gadolinium (III)   1,4,7,10-Tetraazacyclododecane-1,4,7,10-tetraacetate

X-207

Gd-p-SCN-Bn-DOTA

2126179-26-6

Gadolinium (III)   S-2-(4-isothiocyanatobenzyl)-1,4,7,10-tetraazacyclododecane-1,4,7,10-tetraacetic   acid

X-279

Ho-Maleimido-DOTA

1349103-97-4

Holmium (III)   1,4,7,10-tetraazacyclododecane-1,4,7-tris(acetic acid)-_x000D_

10-maleimidoethylacetamide

反應中間體

I-121

Bis-CBZ-Cyclen

162148-45-0

1,4,7,10-Tetraazacyclododecane-1,7-bis(benzylcarbamide)

M-120

DO2A-tert-butyl ester

162148-48-3

1,4,7,10-Tetraazacyclododecane-1,7-bis(t-butyl   acetate)

173308-19-5

2-Aminoethyl-mono-amide-DOTA-tris(t-Bu   ester)

Bifunctional   Chelators (BFCs)-雙分子螯合劑

500 mg/1   g/ 5 g

753421-63-5

4-Aminobutyl-DOTA

Bifunctional   Chelators (BFCs)

100/500   mg

1402393-59-2

4-Aminobutyl-DOTA-tris   (t-butyl ester)

Bifunctional   Chelators (BFCs)

100/500   mg

1227407-76-2

Azido-mono-amide-DOTA

Bifunctional   Chelators (BFCs)

100/500   mg 1g

287970-46-1

EAM-1

Fluorescent Probes

N,N,N-Trimethyl-2[(7-nitro-1,2,3-benzoxadiazol-4-yl)amino]   乙胺碘化物

2125661-97-2

EAM-2

Fluorescent Probes

N,N-二甲基-N-(2-)-2[(7-nitro-1,2,3-benzoxadiazol-4-yl)amino] ethanaminium bromide

2125661-93-8

DO3A-Serotonin

Conjugates（共軛物）

1-(5-Hydroxyindole-3-ethylacetamide)-4,7,10-triaceticacid-1,4,7,10-tetraazacyclododecane

180978-54-5

DOTA-Biotin-Sarcosine

Conjugates

(N-methyl-N-(hexahydro-2-oxo-1H-thieno[3,4-d]-imidazol-4-yl)-oxopentyl)glycyl-2-(S)-(4-aminobenzyl)-1,4,7,10-tetraaceticacid-1,4,7,10-tetraazacyclododecane

177943-89-4

DOTATATE

Conjugates

DOTA-d-Phe-Cys-Tyr-d-Trp-Lys-Thr-Cys-Thr

1/5 mg

130701-19-8

CB-Cyclam

Macrocyclic   Ligands-大環配體

500   mg/1 g

112193-75-6

DO2A

Macrocyclic   Ligands

500   mg/1 g